Antiplasmodial and antileishmanial activities of compounds from Piper tuberculatum Jacq fruits
Abstract INTRODUCTION This study assessed the activity of compounds from Piper tuberculatum against Plasmodium falciparum and Leishmania guyanensis. METHODS The effects of compounds from P. tuberculatum fruits on P. falciparum and L. guyanensis promastigote growth in vitro were determined. Hemolytic...
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ftdoajarticles:oai:doaj.org/article:ccd093f234d64258bf17dd69046beee9 2023-05-15T14:59:34+02:00 Antiplasmodial and antileishmanial activities of compounds from Piper tuberculatum Jacq fruits Flávio Augusto de Souza Oliveira Guilherme Matos Passarini Daniel Sol Sol de Medeiros Ana Paula de Azevedo Santos Saara Neri Fialho Aurileya de Jesus Gouveia Marcinete Latorre Elci Marlei Freitag Patrícia Soares de Maria de Medeiros Carolina Bioni Garcia Teles Valdir Alves Facundo https://doi.org/10.1590/0037-8682-0309-2017 https://doaj.org/article/ccd093f234d64258bf17dd69046beee9 EN eng Sociedade Brasileira de Medicina Tropical (SBMT) http://www.scielo.br/scielo.php?script=sci_arttext&pid=S0037-86822018000300382&lng=en&tlng=en https://doaj.org/toc/1678-9849 1678-9849 doi:10.1590/0037-8682-0309-2017 https://doaj.org/article/ccd093f234d64258bf17dd69046beee9 Revista da Sociedade Brasileira de Medicina Tropical, Vol 51, Iss 3, Pp 382-386 Malaria Leishmaniasis Piper Bioactivity Arctic medicine. Tropical medicine RC955-962 article ftdoajarticles https://doi.org/10.1590/0037-8682-0309-2017 2022-12-31T02:55:15Z Abstract INTRODUCTION This study assessed the activity of compounds from Piper tuberculatum against Plasmodium falciparum and Leishmania guyanensis. METHODS The effects of compounds from P. tuberculatum fruits on P. falciparum and L. guyanensis promastigote growth in vitro were determined. Hemolytic action and cytotoxicity in HepG2 and J774 cells were measured. RESULTS Three compounds showed strong antiplasmodial activity and one compound showed strong antileishmanial activity. Two compounds were non-toxic to HepG2 cells and all were toxic to J774 cells. The compounds showed no hemolytic activity. CONCLUSIONS The tested compounds from P. tuberculatum exhibited antiparasitic and cytotoxic effects. Article in Journal/Newspaper Arctic Directory of Open Access Journals: DOAJ Articles Arctic Revista da Sociedade Brasileira de Medicina Tropical 51 3 382 386 |
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Directory of Open Access Journals: DOAJ Articles |
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English |
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Malaria Leishmaniasis Piper Bioactivity Arctic medicine. Tropical medicine RC955-962 |
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Malaria Leishmaniasis Piper Bioactivity Arctic medicine. Tropical medicine RC955-962 Flávio Augusto de Souza Oliveira Guilherme Matos Passarini Daniel Sol Sol de Medeiros Ana Paula de Azevedo Santos Saara Neri Fialho Aurileya de Jesus Gouveia Marcinete Latorre Elci Marlei Freitag Patrícia Soares de Maria de Medeiros Carolina Bioni Garcia Teles Valdir Alves Facundo Antiplasmodial and antileishmanial activities of compounds from Piper tuberculatum Jacq fruits |
topic_facet |
Malaria Leishmaniasis Piper Bioactivity Arctic medicine. Tropical medicine RC955-962 |
description |
Abstract INTRODUCTION This study assessed the activity of compounds from Piper tuberculatum against Plasmodium falciparum and Leishmania guyanensis. METHODS The effects of compounds from P. tuberculatum fruits on P. falciparum and L. guyanensis promastigote growth in vitro were determined. Hemolytic action and cytotoxicity in HepG2 and J774 cells were measured. RESULTS Three compounds showed strong antiplasmodial activity and one compound showed strong antileishmanial activity. Two compounds were non-toxic to HepG2 cells and all were toxic to J774 cells. The compounds showed no hemolytic activity. CONCLUSIONS The tested compounds from P. tuberculatum exhibited antiparasitic and cytotoxic effects. |
format |
Article in Journal/Newspaper |
author |
Flávio Augusto de Souza Oliveira Guilherme Matos Passarini Daniel Sol Sol de Medeiros Ana Paula de Azevedo Santos Saara Neri Fialho Aurileya de Jesus Gouveia Marcinete Latorre Elci Marlei Freitag Patrícia Soares de Maria de Medeiros Carolina Bioni Garcia Teles Valdir Alves Facundo |
author_facet |
Flávio Augusto de Souza Oliveira Guilherme Matos Passarini Daniel Sol Sol de Medeiros Ana Paula de Azevedo Santos Saara Neri Fialho Aurileya de Jesus Gouveia Marcinete Latorre Elci Marlei Freitag Patrícia Soares de Maria de Medeiros Carolina Bioni Garcia Teles Valdir Alves Facundo |
author_sort |
Flávio Augusto de Souza Oliveira |
title |
Antiplasmodial and antileishmanial activities of compounds from Piper tuberculatum Jacq fruits |
title_short |
Antiplasmodial and antileishmanial activities of compounds from Piper tuberculatum Jacq fruits |
title_full |
Antiplasmodial and antileishmanial activities of compounds from Piper tuberculatum Jacq fruits |
title_fullStr |
Antiplasmodial and antileishmanial activities of compounds from Piper tuberculatum Jacq fruits |
title_full_unstemmed |
Antiplasmodial and antileishmanial activities of compounds from Piper tuberculatum Jacq fruits |
title_sort |
antiplasmodial and antileishmanial activities of compounds from piper tuberculatum jacq fruits |
publisher |
Sociedade Brasileira de Medicina Tropical (SBMT) |
url |
https://doi.org/10.1590/0037-8682-0309-2017 https://doaj.org/article/ccd093f234d64258bf17dd69046beee9 |
geographic |
Arctic |
geographic_facet |
Arctic |
genre |
Arctic |
genre_facet |
Arctic |
op_source |
Revista da Sociedade Brasileira de Medicina Tropical, Vol 51, Iss 3, Pp 382-386 |
op_relation |
http://www.scielo.br/scielo.php?script=sci_arttext&pid=S0037-86822018000300382&lng=en&tlng=en https://doaj.org/toc/1678-9849 1678-9849 doi:10.1590/0037-8682-0309-2017 https://doaj.org/article/ccd093f234d64258bf17dd69046beee9 |
op_doi |
https://doi.org/10.1590/0037-8682-0309-2017 |
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Revista da Sociedade Brasileira de Medicina Tropical |
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51 |
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382 |
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